سيترات الأورفينادرين
| Kind | API |
|---|---|
| Class | Skeletal muscle relaxant — anticholinergic (diphenhydramine analog) |
| Synonyms | Orphenadrini citras |
| Common uses / forms | Tablets and ER tablets (frequently FDC with paracetamol), injection; painful muscle spasm; also antiparkinsonian use |
| Properties | Anticholinergic/antihistaminic with NMDA antagonism; water-soluble citrate salt; well absorbed — BCS Class I; narrow therapeutic index (overdose cardiotoxicity is a clinical caution) |
| Compendia | USP, BP |
| Sourcing origins | EU, India, China |
| Dominant inbound route | Hormuz |
| Indicative price band | $$$ ($100–1000 / kg) |
| Indicative lead time | medium (50–80 days) |
| Notes | Older lower-volume molecule mostly sold as paracetamol FDC; citrate salt distinct from the hydrochloride salt — confirm salt form on order; several but not many qualified sources. |
Open the interactive Data Bank (363 substances) · the full table · Supply Resilience Studio
Share: LinkedIn · X · WhatsApp · Telegram · Email
Cite as: AUPAM Experts' Office, Orphenadrine Citrate — sourcing profile (API) — AUPAM Data Bank, retrieved 2026-08-31, https://aupameo.org/datasets/databank/a-orphenadrine-citrate.html